1 |
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Molecular target interactions of quinoline derivatives as anticancer agents: A review |
Chemical Biology & Drug Design |
101 |
4 |
977-997 |
2023 |
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2 |
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Design, Synthesis, In Vivo, and In Silico Evaluation of Benzothiazoles Bearing a 1, 3, 4-Oxadiazole Moiety as New Antiepileptic Agents |
ACS Omega |
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2023 |
American Chemical Society |
3 |
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Synthesis, Anticonvulsant, and Molecular Docking Studies of (3, 5-disubstituted-4, 5-dihydro-1H-pyrazol-1-yl)(4-chlorophenyl) Methanone Derivatives |
INDIAN JOURNAL OF PHARMACEUTICAL EDUCATION AND RESEARCH |
57 |
1 |
202-209 |
2023 |
ASSOC PHARMACEUTICAL TEACHERS INDIA AL-AMEEN COLL PHARMACY, OPP LALBACH MAIN ⦠|
4 |
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Synthesis Anticonvulsant and Cytotoxic Evaluation of Benzimidazole-Quinoline Hybrids Schiff Base Analogs |
Polycyclic Aromatic Compounds |
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Jan-21 |
2023 |
Taylor & Francis |
5 |
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Conceptual and molecular docking study of newly developed antiepileptic drug cenobamate |
World Journal of Advanced Research and Reviews |
17 |
3 |
281-291 |
2023 |
World Journal of Advanced Research and Reviews |
6 |
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Medicinal and therapeutic properties of Jamun (Syzygium cumini)âA Comprehensive Review |
International Journal of Pharma Professionalâs Research (IJPPR) |
14 |
2 |
15-23 |
2023 |
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7 |
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Synthesis and SAR of Potential Anti-Cancer Agents of Quinoline Analogues: A Review |
Medicinal Chemistry |
19 |
8 |
785-812 |
2023 |
Bentham Science Publishers |
8 |
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Synthesis, Characterization, In Silico and In Vivo Evaluation of BenzimidazoleâBearing Quinoline Schiff Bases as New Anticonvulsant Agents |
ChemistrySelect |
8 |
21 |
e202300209 |
2023 |
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9 |
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Benzimidazole-Quinoline Hybrid Scaffold as Promising Pharmacological Agents: A Review |
Polycyclic Aromatic Compounds |
42 |
8 |
5044-5066 |
2022 |
Taylor & Francis |
10 |
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Recent advances and SAR study of 2-substituted benzothiazole scaffold based potent chemotherapeutic agents |
Results in Chemistry |
4 |
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100258 |
2022 |
Elsevier |
11 |
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Advances of Benzimidazole Derivatives as Anticancer Agents: Bench to Bedside |
Benzimidazole |
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3 |
2022 |
BoDâBooks on Demand |
12 |
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Novel approaches for the development of direct KRAS inhibitors: structural insights and drug design |
Expert Opinion on Drug Discovery |
17 |
3 |
247-257 |
2022 |
Taylor & Francis |
13 |
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An appraisal of anticancer activity with structureâactivity relationship of quinazoline and quinazolinone analogues through EGFR and VEGFR inhibition: A review |
Drug Development Research |
83 |
4 |
859-890 |
2022 |
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14 |
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Design, synthesis, and pharmacological evaluation of aryl oxadiazole linked 1, 2, 4-triazine derivatives as anticonvulsant agents |
Medicinal Chemistry Research |
31 |
5 |
781-793 |
2022 |
Springer US |
15 |
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A comprehensive review on pyrazoline based heterocyclic hybrids as potent anticancer agents |
European Journal of Medicinal Chemistry Reports |
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100042 |
2022 |
Elsevier Masson |
16 |
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Design, synthesis, biological evaluation, and in silico studies of 2âaminobenzothiazole derivatives as potent PI3Kα inhibitors |
Archiv der Pharmazie |
355 |
10 |
2200146 |
2022 |
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17 |
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Combinatorial delivery of Ribociclib and green tea extract mediated nanostructured lipid carrier for oral delivery for the treatment of breast cancer synchronising in silico, in vitro, and in vivo studies |
Journal of Drug Targeting |
30 |
10 |
1113-1134 |
2022 |
Taylor & Francis |
18 |
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Synthesis, biological evaluation, and in silico studies of indoleâtethered pyrazoline derivatives as anticancer agents targeting topoisomerase IIα |
Drug Development Research |
83 |
7 |
1555-1577 |
2022 |
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19 |
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Synthesis, molecular docking, and pharmacological evaluation of 5-(4-(2-(5-ethyl pyridine-2-yl) ethoxy) benzyl)-3-(phenylsulfonyl) thiazolidine-2, 4-dione against HFD-induced diabesity via interaction with the CB1 receptor. |
Iranian Journal of Basic Medical Sciences |
25 |
8 |
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2022 |
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20 |
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Strategies in synthetic design and structureâactivity relationship studies of novel heterocyclic scaffolds as aldose reductaseâ2 inhibitors |
Archiv der Pharmazie |
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e2200167 |
2022 |
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21 |
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Recent Updates on Synthesis, Biological Activity, and Structure-Activity Relationship of 1, 3, 4-oxadiazole-Quinoline Hybrids: A Review. |
Current Organic Synthesis |
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2022 |
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22 |
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Synthesis and Cytotoxic Activity of 1, 2, 4-Triazolo-Linked Bis-Indolyl Conjugates as Dual Inhibitors of Tankyrase and PI3K |
Molecules |
27 |
21 |
7642 |
2022 |
MDPI |
23 |
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Synthesis, Anticonvulsant, and Molecular Docking Studies of 2-(2-Benzyl-1H-benzo [d] imidazol-1-yl)-1-(3, 5-disubstituted phenyl)-4, 5-dihydro-1H-pyrazol-1-yl) ethan-1-ones |
INDIAN JOURNAL OF HETEROCYCLIC CHEMISTRY |
32 |
3 |
321-330 |
2022 |
CONNECT JOURNALS D-189 RAMPRATSHA, PO CHANDER NAGAR, GHAZIABAD, 201 011, INDIA |
24 |
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Synthesis and Pharmacological Evaluation of Some New (1H-Benzimidazol-2-yl)-substituted Methyl-1-(6-substituted-2-chloroquinolin-3-yl) Methanimines |
INDIAN JOURNAL OF HETEROCYCLIC CHEMISTRY |
32 |
3 |
379-385 |
2022 |
CONNECT JOURNALS D-189 RAMPRATSHA, PO CHANDER NAGAR, GHAZIABAD, 201 011, INDIA |
25 |
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Integrated modelling to support analysis of Pandemic Impacts on Roorkee City Water System and Associated Gangatic river water quality. |
AGU Fall Meeting Abstracts |
2022 |
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H15R-1013 |
2022 |
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26 |
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Chitosan coated synergistically engineered nanoemulsion of Ropinirole and nigella oil in the management of Parkinson's disease: Formulation perspective and In vitro and In vivo assessment |
International Journal of Biological Macromolecules |
167 |
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605-619 |
2021 |
Elsevier |
27 |
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Synthesis and anticonvulsant evaluation of indoline derivatives of functionalized aryloxadiazole amine and benzothiazole acetamide |
Journal of Molecular Structure |
1228 |
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129742 |
2021 |
Elsevier |
28 |
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Design, in-silico study and biological evaluation of newly synthesized 3-chlorobenzofuran congeners as antitubercular agents |
Arabian Journal of Chemistry |
14 |
4 |
103034 |
2021 |
Elsevier |
29 |
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Roflumilast and tadalafil improve learning and memory deficits in intracerebroventricular Aβ1â42 rat model of Alzheimerâs disease through modulations of hippocampal cAMP/cGMP/BDNF signaling pathway |
Pharmacological Reports |
73 |
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1287-1302 |
2021 |
Springer International Publishing |
30 |
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1, 3, 4-oxadiazoles as potential pharmacophore for cytotoxic potentiality: a comprehensive review |
Current Topics in Medicinal Chemistry |
21 |
15 |
1377-1397 |
2021 |
Bentham Science Publishers |
31 |
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Advances in 2âsubstituted benzothiazole scaffoldâbased chemotherapeutic agents |
Archiv der Pharmazie |
354 |
12 |
2100246 |
2021 |
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32 |
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Pharmacophore based drug design and synthesis of oxindole bearing hybrid as anticancer agents |
Bioorganic Chemistry |
116 |
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105358 |
2021 |
Academic Press |
33 |
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Insight into the Isolation, Synthesis, and Structure-Activity Relationship of Piperine Derivatives for the Development of New Compounds: Recent Updates |
Current Topics in Medicinal Chemistry |
21 |
30 |
2715-2751 |
2021 |
Bentham Science Publishers |
34 |
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The Synthesis and Anticancer Potentials of Quinoline Analogues: A Review of Literature |
Mini-Reviews in Organic Chemistry |
18 |
6 |
735-768 |
2021 |
Bentham Science Publishers |
35 |
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Apoptosis Inducing 1, 3, 4-Oxadiazole Conjugates of Capsaicin: Their In Vitro Antiproliferative and In Silico Studies |
ACS Medicinal Chemistry Letters |
12 |
11 |
1694-1702 |
2021 |
American Chemical Society |
36 |
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Synthesis, Characterization, and Antidiabetic Evaluation of Substituted 5-(2-Chloro-Quinolin-3-Ylmethylene)-Thiazolidine-2, 4-Dione |
J. Heterocycl. Chem |
31 |
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01-Aug |
2021 |
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37 |
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Integrated Modelling to Support Analysis of COVID-19 Impacts on Haridwars City Water System and Ganga river water quality. |
AGU Fall Meeting Abstracts |
2021 |
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GH15F-0637 |
2021 |
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38 |
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SARS-CoV-2: Molecular Biology and Therapeutic Targets |
Coronaviruses |
2 |
11 |
May-19 |
2021 |
Bentham Science Publishers |
39 |
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Recent progress of Benzimidazole hybrids for anticancer potential |
Current Medicinal Chemistry |
27 |
35 |
5970-6014 |
2020 |
Bentham Science Publishers |
40 |
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Neurological and psychiatric management using COMT inhibitors: A review |
Bioorganic chemistry |
94 |
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103418 |
2020 |
Academic Press |
41 |
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Design and synthesis of newer 1, 3, 4-oxadiazole and 1, 2, 4-triazole based Topsentin analogues as anti-proliferative agent targeting tubulin |
Bioorganic chemistry |
95 |
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103519 |
2020 |
Academic Press |
42 |
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Synthesis, anti-convulsant activity and molecular docking study of novel thiazole pyridazinone hybrid analogues |
Bioorganic chemistry |
99 |
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103584 |
2020 |
Academic Press |
43 |
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Molecular interactions of vinclozolin metabolites with human estrogen receptors 1GWR-α and 1QKM and androgen receptor 2AM9-β: Implication for endocrine disruption |
Toxicology Mechanisms and Methods |
30 |
5 |
370-377 |
2020 |
Taylor & Francis |
44 |
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Synthetic lethality on drug discovery: an update on cancer therapy |
Expert Opinion on Drug Discovery |
15 |
7 |
823-832 |
2020 |
Taylor & Francis |
45 |
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Aromatase inhibitors: Role in postmenopausal breast cancer |
Archiv Der Pharmazie |
353 |
8 |
2000081 |
2020 |
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46 |
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Free radical scavengers: An overview on heterocyclic advances and medicinal prospects |
European Journal of Medicinal Chemistry |
204 |
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112607 |
2020 |
Elsevier Masson |
47 |
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Synthesis, antimicrobial, and molecular docking studies of 1,3-Thiazolidin-4-one analogs bearing benzothiazole |
Indian Journal of Heterocyclic Chemistry |
30 |
2 |
325-335 |
2020 |
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48 |
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Clinical Trial: The Most Critical Step in the Process of Drug Development |
Biosciences Biotechnology Research Asia |
3 |
2 (a) |
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2020 |
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49 |
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Anti-tubulin agents of natural origin: Targeting taxol, vinca, and colchicine binding domains |
European journal of medicinal chemistry |
171 |
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310-331 |
2019 |
Elsevier Masson |
50 |
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Correction to: Substituted phenyl containing 1, 3, 4-oxadiazole-2-yl-but-2-enamides: synthesis and preliminary evaluation as promising anticonvulsants |
Medicinal Chemistry Research |
28 |
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926-926 |
2019 |
Springer US |
51 |
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Novel 9-(2-(1-arylethylidene) hydrazinyl) acridine derivatives: Target Topoisomerase 1 and growth inhibition of HeLa cancer cells |
Bioorganic chemistry |
88 |
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102962 |
2019 |
Academic Press |
52 |
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Medicinal prospects of antioxidants: A review |
European journal of medicinal chemistry |
178 |
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687-704 |
2019 |
Elsevier Masson |
53 |
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Synthesis and Biological Potentials of Quinoline Analogues: Review of Literature |
Mini Reviews in Organic Chemistry |
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2019 |
Bentham Science |
54 |
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Tubulin inhibitors as novel anticancer agents: an overview on patents (2013-2018) |
Expert opinion on therapeutic patents |
29 |
8 |
623-641 |
2019 |
Taylor & Francis |
55 |
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Anticonvulsant evaluation of 2-pyrazolines carrying naphthyl moiety: An insight into synthesis and molecular docking study |
Brazilian Journal of Pharmaceutical Sciences |
55 |
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2019 |
Universidade de São Paulo, Faculdade de Ciências Farmacêuticas |
56 |
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Synthetic strategy and SAR studies of C-glucoside heteroaryls as SGLT2 inhibitor: A review |
European journal of medicinal chemistry |
184 |
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111773 |
2019 |
Elsevier Masson |
57 |
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Design and synthesis of cell selective α/β-diastereomeric peptidomimetic with potent in vivo antibacterial activity against methicillin resistant S. aureus |
Bioorganic Chemistry |
76 |
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538-547 |
2018 |
Academic Press |
58 |
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Pyridazinone hybrids: Design, synthesis and evaluation as potential anticonvulsant agents |
Bioorganic Chemistry |
77 |
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74-83 |
2018 |
Academic Press |
59 |
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High-salt-and cholesterol diet-associated cognitive impairment attenuated by tannins-enriched fraction of Emblica officinalis via inhibiting NF-kB pathway |
Inflammopharmacology |
26 |
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147-156 |
2018 |
Springer International Publishing |
60 |
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Rosuvastatin ameliorates cognitive impairment in rats fed with high-salt and cholesterol diet via inhibiting acetylcholinesterase activity and amyloid beta peptide aggregation |
Human & Experimental Toxicology |
37 |
4 |
399-411 |
2018 |
SAGE Publications Sage UK: London, England |
61 |
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Synthesis of stable benzimidazole derivatives bearing pyrazole as anticancer and EGFR receptor inhibitors |
Bioorganic Chemistry |
78 |
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158-169 |
2018 |
Academic Press |
62 |
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Current perspectives on quinazolines with potent biological activities: A review |
Synthetic Communications |
48 |
10 |
1099-1127 |
2018 |
Taylor & Francis |
63 |
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1, 2, 3-triazole tethered Indole-3-glyoxamide derivatives as multiple inhibitors of 5-LOX, COX-2 & tubulin: Their anti-proliferative & anti-inflammatory activity |
Bioorganic chemistry |
81 |
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Jan-20 |
2018 |
Academic Press |
64 |
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DYRK1A kinase inhibition with emphasis on neurodegeneration: A comprehensive evolution story-cum-perspective |
European Journal of Medicinal Chemistry |
158 |
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559-592 |
2018 |
Elsevier Masson |
65 |
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Emergence of promising novel DPPâ4 inhibitory heterocycles as antiâdiabetic agents: A review |
Archiv Der Pharmazie |
351 |
8 |
Jan-14 |
2018 |
WILEY-VCH Verlag GmbH & Co. KGaA, Weinheim |
66 |
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Novel fluoroquinolone derivatives bearing N-thiomide linkage with 6-substituted-2-aminobenzothiazoles: synthesis and antibacterial evaluation |
Arabian Journal of Chemistry |
10 |
1 |
S568-S575 |
2017 |
Elsevier |
67 |
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Synthesis, characterization and antimicrobial activity of 1, 3, 4-oxadiazole bearing 1H-benzimidazole derivatives |
Arabian Journal of Chemistry |
10 |
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S503âS508 |
2017 |
Elsevier |
68 |
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Establishment of inherent stability on piracetam by UPLC/HPLC and development of a validated stability-indicating method |
Arabian Journal of Chemistry |
10 |
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S576âS582 |
2017 |
Elsevier |
69 |
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Structure-activity relationship (SAR) study and design strategies of nitrogen-containing heterocyclic moieties for their anticancer activities |
European journal of medicinal chemistry |
125 |
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143-189 |
2017 |
Elsevier Masson |
70 |
|
Synthesis, characterization and antimicrobial activity of 1, 3, 4-oxadiazole bearing 1H-benzimidazole derivatives |
Arabian Journal of Chemistry |
10 |
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S503-S508 |
2017 |
Elsevier |
71 |
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Recent advances in the synthesis and anticancer activity of molecules other than nitrogen containing heterocyclic moeities. |
Mini reviews in medicinal chemistry |
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2017 |
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72 |
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In vivo anti-inflammatory activity and docking study of newly synthesized benzimidazole derivatives bearing oxadiazole and morpholine rings |
Bioorganic Chemistry |
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2017 |
Academic Press |
73 |
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Design, synthesis, docking and QSAR study of substituted benzimidazole linked oxadiazole as cytotoxic agents, EGFR and erbB2 receptor inhibitors |
European Journal of Medicinal Chemistry |
126 |
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853-869 |
2017 |
Elsevier Masson |
74 |
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Quinazolines and Anticancer Activity: A Current Perspectives |
Synthetic Communications |
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47 (5), 379-408 |
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2017 |
Taylor & Francis |
75 |
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Design, synthesis, and biological evaluation of novel quinazoline clubbed thiazoline derivatives |
Archiv der Pharmazie |
350 |
2 |
1600298 |
2017 |
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76 |
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Design and synthesis of quinazoline-3, 4-(4H)-diamine endowed with thiazoline moiety as new class for DPP-4 and DPPH inhibitor |
Bioorganic Chemistry |
71 |
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181-191 |
2017 |
Academic Press |
77 |
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Benzimidazoles: A biologically active compounds |
Arabian Journal of Chemistry |
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10 |
S157âS173 |
2017 |
Elsevier |
78 |
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Design, synthesis, anticonvulsant evaluation and docking study of 2-[(6-substituted benzo [d] thiazol-2-ylcarbamoyl) methyl]-1-(4-substituted phenyl) isothioureas |
Bioorganic Chemistry |
71 |
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230-243 |
2017 |
Academic Press |
79 |
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Design, synthesis and anticonvulsant evaluation of N-[(substituted 1H-pyrazol-3-yl) amino]-2-(4-methylphenyl) quinazolin-4 (3H)-one derivatives |
Asian J Chem |
29 |
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1375-1379 |
2017 |
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80 |
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Design, synthesis, and docking study of pyrimidineâtriazine hybrids for GABA estimation in animal epilepsy models |
Archiv der Pharmazie |
350 |
9 |
1700146 |
2017 |
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81 |
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Updates on synthesis and biological activities of 1, 3, 4-oxadiazole: A review |
Synthetic Communications |
47 |
20 |
1805-1847 |
2017 |
Taylor & Francis |
82 |
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Design, synthesis, and pharmacological screening of pyridazinone hybrids as anticonvulsant agents |
Archiv der Pharmazie |
350 |
10 |
1700135 |
2017 |
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83 |
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Synthesis and anticonvulsant activity of a combined pharmacophore of 2-oxo-1, 2-dihydroquinoline containing 1, 3, 4-oxadiazole derivatives |
Indian Journal of Heterocyclic Chemistry |
27 |
1 |
33-41 |
2017 |
Connect Journals |
84 |
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Determination of novel phase I metabolite of febuxostat followed by In Vitro, In Vivo Pharmacokinetic and In Silico Studies |
EC Pharmacology and Toxicology |
4 |
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120-134 |
2017 |
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85 |
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Synthesis, characterization and pharmacological screening of novel benzimidazole derivatives |
Arabian Journal of Chemistry |
9 |
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S342-S347 |
2016 |
Elsevier |
86 |
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Design, synthesis, and biological evaluation of 6â(2âaminoâsubstituted phenyl)â4â(substituted phenyl)â1, 2, 4âtriazineâ3, 5 (2H, 4H)âdione derivatives as anticonvulsant agents |
Archiv der Pharmazie |
349 |
4 |
277-292 |
2016 |
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87 |
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Antidepressant, analgesic activity and SAR studies of substituted benzimidazoles |
Asian Journal of Pharmaceutical Research |
6 |
3 |
170-174 |
2016 |
A & V Publications |
88 |
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Synthesis of new benzimidazole and phenylhydrazinecarbothiomide hybrids and their anticonvulsant activity |
Medicinal Chemistry Research |
25 |
7 |
1390â1402 |
2016 |
Springer |
89 |
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Physicochemical characterization of benzalkonium chloride and urea based deep eutectic solvent (DES): A novel catalyst for the efficient synthesis of isoxazolines under ultrasonic irradiation |
Journal of Molecular Liquids |
224 |
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1249-1255 |
2016 |
Elsevier |
90 |
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Tacrolimus-loaded nanostructured lipid carriers for oral delivery-in vivo bioavailability enhancement |
European Journal of Pharmaceutics and Biopharmaceutics |
109 |
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European Journal of Pharmaceutics and Bi |
2016 |
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91 |
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Tacrolimus-loaded nanostructured lipid carriers for oral delivery â Optimization of production and characterization |
European Journal of Pharmaceutics and Biopharmaceutics |
108 |
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277-288 |
2016 |
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92 |
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Self assembly and hydrogelation of spermine functionalized aromatic peptidomimetics against planktonic and sessile methicillin resistant S. aureus |
RSC advances |
6 |
113 |
112656-112666 |
2016 |
Royal Society of Chemistry |
93 |
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Synthesis and antibacterial evaluation of novel analogs of fluoroquinolones annulated with 6-substituted-2-aminobenzothiazoles |
Arabian Journal of Chemistry |
8 |
5 |
671-677 |
2015 |
Elsevier |
94 |
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Design, synthesis, and biological evaluation of thiazolidineâ2, 4âdione conjugates as PPARâγ agonists |
Archiv der Pharmazie |
348 |
6 |
421-432 |
2015 |
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95 |
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Synthesis and evaluation of benzimidazole derivatives as selective COX-2 inhibitors |
Medicinal Chemistry |
11 |
2 |
188-199 |
2015 |
Bentham Science Publishers |
96 |
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Synthesis, antibacterial and anticancer evaluation of 5-substituted (1, 3, 4-oxadiazol-2-yl) quinoline |
Medicinal Chemistry Research |
24 |
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2514-2528 |
2015 |
Springer US |
97 |
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N-terminal aromatic tag induced self assembly of tryptophanâarginine rich ultra short sequences and their potent antibacterial activity |
RSC advances |
5 |
84 |
68610-68620 |
2015 |
Royal Society of Chemistry |
98 |
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Design, synthesis, in silico molecular docking and biological evaluation of novel oxadiazole based thiazolidine-2, 4-diones bis-heterocycles as PPAR-γ agonists |
European Journal of Medicinal Chemistry |
87 |
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175-185 |
2014 |
Elsevier Masson |
99 |
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Thiazolidine-2, 4-diones derivatives as PPAR-γ agonists: Synthesis, molecular docking, in vitro and in vivo antidiabetic activity with hepatotoxicity risk evaluation and effect on PPAR-γ gene expression |
Bioorganic & medicinal chemistry letters |
24 |
14 |
3034-3042 |
2014 |
Elsevier |
100 |
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Substituted phenyl containing 1, 3, 4-oxadiazole-2-yl-but-2-enamides: synthesis and preliminary evaluation as promising anticonvulsants |
Medicinal Chemistry Research |
23 |
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4915-4925 |
2014 |
Springer US |
101 |
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Design, synthesis and docking studies of 2-benzoxazolinone-based 1, 2, 4-triazoles as proinflammatory cytokine inhibitors |
Medicinal Chemistry Research |
23 |
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4250-4268 |
2014 |
Springer US |
102 |
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Synthesis, characterization and biological evaluation of novel 1, 2, 4-triazole derivatives as potent antibacterial and anti-inflammatory agents |
Der Pharma Chemica |
6 |
1 |
137-43 |
2014 |
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103 |
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Synthesis, characterization and anticancer evaluation of 2-(naphthalen-1-ylmethyl/naphthalen-2-yloxymethyl)-1-[5-(substituted phenyl)-[1, 3, 4] oxadiazol-2-ylmethyl]-1H-benzimidazole |
Arabian Journal of Chemistry |
7 |
4 |
418-424 |
2014 |
Elsevier |
104 |
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Synthesis, characterization, and in vitro anticancer evaluation of novel 2, 5-disubstituted 1, 3, 4-oxadiazole analogue |
BioMed research international |
2014 |
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2014 |
Hindawi |
105 |
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Synthesis, biological activities, and pharmacokinetics studies of a mutual prodrug of aceclofenac and paracetamol |
Medicinal Chemistry Research |
23 |
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1077-1083 |
2014 |
Springer US |
106 |
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Anticancer activity of new compounds using benzimidazole as a scaffold |
Anti-Cancer Agents in Medicinal Chemistry (Formerly Current Medicinal Chemistry-Anti-Cancer Agents) |
14 |
7 |
1003-1018 |
2014 |
Bentham Science Publishers |
107 |
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Design and synthesis of benzimidazole analogs endowed with oxadiazole as selective COXâ2 inhibitor |
Archiv der Pharmazie |
347 |
12 |
923-935 |
2014 |
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108 |
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Design and synthesis of pyrimidine molecules endowed with thiazolidin-4-one as new anticancer agents |
European journal of medicinal chemistry |
83 |
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630-645 |
2014 |
Elsevier |
109 |
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Synthesis and antihypertensive screening of new derivatives of quinazolines linked with isoxazole |
BioMed Research International |
2014 |
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2014 |
Hindawi |
110 |
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Pharmacokinetic interaction between febuxostat and morin in rats |
Expert Opinion on Drug Metabolism & Toxicology |
10 |
3 |
307-312 |
2014 |
Taylor & Francis |
111 |
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Synthesis and characterization of quinazoline derivatives: search for hybrid molecule as diuretic and antihypertensive agents |
Journal of Enzyme Inhibition and Medicinal Chemistry |
29 |
5 |
733-743 |
2014 |
Taylor & Francis |
112 |
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Isolation, identification and characterization of degradation product of piracetam using analytical techniques |
IJARSC |
7 |
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Aug-16 |
2014 |
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113 |
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N-terminally modified linear and branched spermine backbone dipeptidomimetics against planktonic and sessile methicillin-resistant Staphylococcus aureus |
Antimicrobial Agents and Chemotherapy |
58 |
9 |
5435-5447 |
2014 |
American Society for Microbiology 1752 N St., NW, Washington, DC |
114 |
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The impact of internal marketing on the employee's retention in Sialkot industries |
International Journal of Academic Research in Business and Social Sciences |
4 |
9 |
478 |
2014 |
Human Resource Management Academic Research Society |
115 |
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Salahuddin, Mohammad Shaharyar b, Avijit Mazumder |
Arabian Journal of Chemistry |
7 |
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418-424 |
2014 |
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116 |
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Microwave assisted one pot synthesis of some pyrazole derivatives as a safer anti-inflammatory and analgesic agents |
Acta Pol. Pharm |
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Synthesis and Biological Evaluation of Some Novel Oxadiazoles Derived from Bi phenyl 4-carboxylic acid. |
Der Pharmacia Lettre |
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Analytical methods for the detection of undeclared synthetic drugs in traditional herbal medicines as adulterants |
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Application of LCâMS/MS for quantitative analysis of glucocorticoids and stimulants in biological fluids |
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Elsevier |
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Benzimidazole clubbed with triazolo-thiadiazoles and triazolo-thiadiazines: New anticancer agents |
European journal of medicinal chemistry |
62 |
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Elsevier Masson |
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Establishment of inherent stability of febuxostat and development of a validated stability-indicating method by UPLC according to ICH requirement |
Medicinal Chemistry Research |
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Springer-Verlag |
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Chromatographic separation of piracetam and its metabolite in a mixture of microsomal preparations, followed by an MS/MS analysis |
European journal of medicinal chemistry |
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Elsevier Masson |
126 |
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Molecular properties prediction, synthesis, and diuretic activity of phenoxy acetic acid bearing pyrazolines |
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Springer-Verlag |
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Design, Synthesis, and Biological Evaluation of 6-(2-Amino-substituted phenyl)-4-(substituted phenyl)-1,2,4-triazine-3,5(2H,4H)-dione Derivatives as Anticonvulsant Agents |
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WILEYâVCH Verlag Weinheim |
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Comparative study of forced degradation behavior of telmisartan by UPLC and HPLC and development of validated stability indicating assay method according to ICH guidelines |
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Synthesis of quinoline attached-furan-2 (3H)-ones having anti-inflammatory and antibacterial properties with reduced gastro-intestinal toxicity and lipid peroxidation |
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Synthesis and in vivo diuretic activity of some novel pyrimidine derivatives |
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Taylor & Francis |
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Synthesis of novel 8-hydroxy quinolin based 1, 3, 4-oxadiazoles and S-substituted 1, 2, 4-triazole derivatives and evaluation of their anti-inflammatory, analgesic, ulcerogenic and anti-microbial activities |
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Bentham Science Publishers |
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Triazole incorporated pyridazinones as a new class of antihypertensive agents: Design, synthesis and in vivo screening |
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Recent advances and future perspectives of triazole analogs as promising antiviral agents |
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Bentham Science Publishers |
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Current medicinal chemistry |
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Curr. Med. Chem |
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26 |
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142 |
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Therapeutic importance of peptidomimetics in medicinal chemistry |
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Molecular properties prediction, synthesis and antimicrobial activity of some newer oxadiazole derivatives |
European journal of medicinal chemistry |
45 |
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Elsevier Masson |
144 |
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Ciprofloxacin: review on developments in synthetic, analytical, and medicinal aspects |
Journal of enzyme inhibition and medicinal chemistry |
25 |
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Taylor & Francis |
145 |
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Simultaneous estimation of simvastatin and ezetimibe in pharmaceutical tablet dosage forms by RP-HPLC: A Review |
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Pyrazoline bearing benzimidazoles: search for anticancer agent |
European journal of medicinal chemistry |
45 |
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European journal of medicinal chemistry |
45 |
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151 |
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Antimicrobial activities of some synthetic butenolides and their pyrrolone derivatives |
Journal of Enzyme Inhibition and Medicinal Chemistry |
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Taylor & Francis |
152 |
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Microwave assisted synthesis, characterization & biological evaluation of benzimidazole substituted 1, 3, 4-oxadiazole |
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Synthesis and Evaluation of Pyrrole Derivative Conjugates of Aspirin as Anti-Platelet Agents |
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Chemical Investigation of Polygonatum verticillatum |
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Clinical profile and risk factors in late hemorrhagic disease of newborn: our experience |
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Synthesis and in vivo diuretic activity of biphenyl benzothiazole-2-carboxamide derivatives |
Acta Pol Pharm Drug Res |
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World Acad. Sci. Engr. Tech |
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Design, synthesis and evaluation of novel 5, 6-dimethoxy-1-oxo-2, 3-dihydro-1H-2-indenyl-3, 4-substituted phenyl methanone analogues |
Bioorganic & medicinal chemistry letters |
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Acta Poloniae Pharmaceutica-Drug Research |
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Synthesis and evaluation of in vitro antiviral activity of novel phenoxy acetic acid derivatives |
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Microwave Assisted Synthesis, Characterization and Pharmacological Evaluation of Pyridazinone Derivatives |
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Synthesis and antihyperglycemic activity of 2-(substituted phenyl)-3-{[4-(1-naphthyl)-1, 3-thiazol-2-yl] amino}-4-oxo-1, 3-thiazolidin-5-ylacetic acid derivatives. |
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Asian Journal of Chemistry |
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Synthesis, antimycobacterial activity of 4-[5-(substituted phenyl)-4, 5-dihydro-3-isoxazolyl]-2-methylphenol |
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Taylor & Francis |
178 |
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Synthesis, characterization and biological studies of novel imines and azetidinones derivatives of haloaryloxy moiety |
Asian Journal of Chemistry |
20 |
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179 |
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Synthesis, characterization and biological studies of new schiff bases and azetidinones derived from propionic acid derivatives |
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Synthesis of novel substituted pyrazolyl-2-toluidinomethanethione and pyrazolyl-2-methoxyanilinomethanethione as potential antitubercular agents |
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SP Birkhäuser Verlag Boston |
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Pergamon |
190 |
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Discovery of novel phenoxyacetic acid derivatives as antimycobacterial agents |
Bioorganic & medicinal chemistry |
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Synthesis and antiproliferative activity of 1-[(sub)]-6-fluoro-3-[(sub)]-1, 3, 4-oxadiazol-2-yl-7-piperazino-1, 4-dihydro-4-quinolinone derivatives |
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Journal of Enzyme Inhibition and Medicinal Chemistry |
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Taylor & Francis |
193 |
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Synthesis, structural activity relationship and anti-tubercular activity of novel pyrazoline derivatives |
European journal of medicinal chemistry |
42 |
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Elsevier Masson |
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Synthesis and anti-HIV activity of N'-nicotinoyl-3-(4'-hydroxy-3'-methylphenyl)-5-[substituted phenyl]-2-pyrazo-lines |
Acta Pol Pharm |
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Acta Pol. Pharm. Drug Res |
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Synthesis and antimycobacterial activity of novel heterocycles |
Journal of the Serbian Chemical Society |
72 |
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Synthesis and cytotoxic activity of novel pyrazoline derivatives against human lung tumor cell line (A549) |
Journal of the Chinese Chemical Society |
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WILEYâVCH Verlag Weinheim |
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Bioorganic & medicinal chemistry letters |
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Elsevier |
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Bioorganic & medicinal chemistry letters |
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Pergamon |
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Design of targeted dosage form of ofloxacin. |
Journal of the Serbian Chemical Society |
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An overview of patents |
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Synthesis and antibacterial activity of epoxides derived from chalcones |
Asian Journal of Chemistry |
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High Throughput Screening As a Versatile Technique of Drug Discovery |
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Recent Updates on Antimicrobial Potential of Novel Oxadiazole Derivatives |
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Synthesis, Characterization and Antimicrobial Activity of New Triazole Derivatives Containing Imidazole Nucleus |
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Synthesis, Characterization and Anti-microbial Activities of 1, 2, 4-Ttriazole & 1, 3, 4-Thiadiazole derivatives of biphenyl-4-carboxylic acid |
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Advances of Benzimidazole Derivatives as Anticancer Agents: Bench to Bedside |
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Global uses of traditional herbs for hepatic diseases and other pharmacological actions: A comprehensive review |
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